Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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EPHA1

RBC: EPHA1 · Substrate: pEY + Mn · high confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Dasatinib98.90.70
Repotrectinib95.20.61
Fostamatinib92.80.61
Crizotinib87.00.58
Erdafitinib86.20.74
Ponatinib75.90.53
Gilteritinib74.20.51
Vandetanib70.00.72
Cabozantinib60.80.75
Pacritinib60.00.45
Nilotinib54.20.77
Regorafenib50.90.72
Dacomitinib49.20.66
Afatinib47.40.71
Ripretinib44.60.67

Known variants

No variants catalogued.
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