Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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FER

RBC: FER · Substrate: pEY · high confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Ceritinib98.40.62
Brigatinib98.20.51
Lorlatinib98.10.69
Lazertinib97.70.67
Repotrectinib96.60.61
Crizotinib94.00.58
Entrectinib91.50.67
Gilteritinib91.00.51
Pacritinib90.40.45
Defactinib84.70.45
Nintedanib83.80.61
Neratinib79.40.60
Alectinib72.70.65
Fostamatinib69.20.61
Sunitinib57.30.52

Known variants

No variants catalogued.
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