GRK6
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Repotrectinib | 44.1 | 0.61 |
| Lorlatinib | 42.0 | 0.69 |
| Midostaurin | 38.0 | 0.50 |
| Sunitinib | 26.1 | 0.52 |
| Capivasertib | 22.4 | 0.64 |
| Nintedanib | 21.6 | 0.61 |
| Ceritinib | 19.6 | 0.62 |
| Larotrectinib | 19.2 | 0.71 |
| Defactinib | 18.7 | 0.45 |
| Cobimetinib | 18.1 | 0.64 |
| Abrocitinib | 15.8 | 0.58 |
| Tivozanib | 15.8 | 0.67 |
| Pirtobrutinib | 14.9 | 0.66 |
| Gedatolisib | 14.2 | 0.61 |
| Mitapivat | 13.8 | 0.63 |
Known variants
No variants catalogued.