Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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GSK3A

RBC: GSK3a · Substrate: Phospho-Glycogen Synthase peptide · medium confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Abemaciclib97.20.56
Defactinib84.10.45
Pacritinib67.40.45
Midostaurin60.70.50
Vemurafenib46.00.60
Encorafenib44.80.76
Pralsetinib42.00.64
Darovasertib36.40.72
Dabrafenib31.70.63
Neratinib30.50.60
Gefitinib27.90.65
Dacomitinib27.50.66
Nintedanib26.80.61
Fostamatinib25.70.61
Imatinib25.00.72

Known variants

No variants catalogued.
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