INSR
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Ceritinib | 97.8 | 0.62 |
| Gilteritinib | 95.1 | 0.51 |
| Brigatinib | 94.0 | 0.51 |
| Alectinib | 91.1 | 0.65 |
| Nintedanib | 90.5 | 0.61 |
| Crizotinib | 89.9 | 0.58 |
| Neratinib | 81.0 | 0.60 |
| Repotrectinib | 72.4 | 0.61 |
| Entrectinib | 72.0 | 0.67 |
| Sunitinib | 71.7 | 0.52 |
| Fostamatinib | 70.9 | 0.61 |
| Pacritinib | 60.6 | 0.45 |
| Bosutinib | 51.5 | 0.55 |
| Defactinib | 48.0 | 0.45 |
| Lorlatinib | 39.0 | 0.69 |
Known variants
No variants catalogued.