IRAK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Pacritinib | 99.6 | 0.45 |
| Abemaciclib | 98.3 | 0.56 |
| Ponatinib | 97.7 | 0.53 |
| Encorafenib | 97.5 | 0.76 |
| Crizotinib | 90.6 | 0.58 |
| Alectinib | 85.2 | 0.65 |
| Tepotinib | 72.6 | 0.73 |
| Afatinib | 72.1 | 0.71 |
| Sunitinib | 71.9 | 0.52 |
| Gilteritinib | 70.2 | 0.51 |
| Brigatinib | 62.9 | 0.51 |
| Gefitinib | 62.4 | 0.65 |
| Dacomitinib | 60.2 | 0.66 |
| Pirtobrutinib | 50.1 | 0.66 |
| Defactinib | 50.0 | 0.45 |
Known variants
No variants catalogued.