ITK
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Canertinib | 96.9 | 0.67 |
| Ibrutinib | 94.5 | 0.72 |
| Mobocertinib | 94.4 | 0.76 |
| Repotrectinib | 88.0 | 0.61 |
| Osimertinib | 85.4 | 0.73 |
| Lazertinib | 84.0 | 0.67 |
| Neratinib | 78.4 | 0.60 |
| Zanubrutinib | 74.5 | 0.79 |
| Dacomitinib | 73.6 | 0.66 |
| Entrectinib | 68.4 | 0.67 |
| Afatinib | 58.7 | 0.71 |
| Nintedanib | 51.9 | 0.61 |
| Ponatinib | 38.8 | 0.53 |
| Brigatinib | 36.6 | 0.51 |
| Sunitinib | 35.2 | 0.52 |
Known variants
No variants catalogued.