JAK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Pralsetinib | 99.1 | 0.64 |
| Abrocitinib | 98.7 | 0.58 |
| Baricitinib | 98.1 | 0.62 |
| Ponatinib | 98.0 | 0.53 |
| Upadacitinib | 97.3 | 0.66 |
| Repotrectinib | 96.9 | 0.61 |
| Ruxolitinib | 96.7 | 0.59 |
| Tenalisib | 96.4 | 0.70 |
| Umbralisib | 96.4 | 0.67 |
| Ripretinib | 96.0 | 0.67 |
| Tofacitinib | 95.2 | 0.68 |
| Fedratinib | 94.2 | 0.58 |
| Defactinib | 93.7 | 0.45 |
| Entrectinib | 93.3 | 0.67 |
| Tucatinib | 92.7 | 0.65 |
Known variants
No variants catalogued.