Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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JAK3

RBC: JAK3 · Substrate: JAK3tide ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Midostaurin100.00.50
Ponatinib99.30.53
Ruxolitinib99.20.59
Canertinib98.90.67
Ibrutinib98.60.72
Tofacitinib98.20.68
Pralsetinib98.10.64
Lazertinib97.70.67
Osimertinib97.50.73
Upadacitinib97.50.66
Mobocertinib97.20.76
Baricitinib97.00.62
Repotrectinib96.20.61
Nintedanib95.20.61
Neratinib95.20.60

Known variants

No variants catalogued.
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