Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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MAP2K7

RBC: MKK7 · Substrate: JNK (K55M) ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Ibrutinib94.80.72
Lazertinib93.80.67
Canertinib80.60.67
Futibatinib60.40.72
Pemigatinib20.10.72
Ponatinib15.40.53
Alpelisib12.80.72
Zanubrutinib12.40.79
Pralsetinib8.70.64
Fedratinib8.50.58
Capmatinib8.40.58
Ripretinib8.10.67
Mitapivat7.30.63
Neratinib7.10.60
Pexidartinib5.00.63

Known variants

No variants catalogued.
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