MAPK8
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Pacritinib | 88.5 | 0.45 |
| Ripretinib | 88.5 | 0.67 |
| Neratinib | 85.7 | 0.60 |
| Brigatinib | 81.8 | 0.51 |
| Fostamatinib | 74.7 | 0.61 |
| Gilteritinib | 73.9 | 0.51 |
| Vemurafenib | 73.8 | 0.60 |
| Encorafenib | 69.9 | 0.76 |
| Fedratinib | 67.8 | 0.58 |
| Abemaciclib | 64.8 | 0.56 |
| Pazopanib | 60.5 | 0.67 |
| Nilotinib | 57.6 | 0.77 |
| Umbralisib | 43.1 | 0.67 |
| Apatinib | 42.7 | 0.70 |
| Dabrafenib | 36.3 | 0.63 |
Known variants
No variants catalogued.