Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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PEAK1

RBC: PEAK1 · Substrate: pEY · high confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Dasatinib99.90.70
Bosutinib97.70.55
Nintedanib94.70.61
Vandetanib94.40.72
Gilteritinib94.00.51
Fostamatinib83.20.61
Brigatinib82.90.51
Midostaurin75.30.50
Dacomitinib75.20.66
Sunitinib73.60.52
Vemurafenib69.70.60
Ibrutinib62.60.72
Pazopanib62.30.67
Afatinib59.80.71
Cabozantinib53.20.75

Known variants

No variants catalogued.
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