PLK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Brigatinib | 58.8 | 0.51 |
| Defactinib | 48.9 | 0.45 |
| Palbociclib | 38.9 | 0.67 |
| Ceritinib | 35.9 | 0.62 |
| Fedratinib | 20.2 | 0.58 |
| Pacritinib | 14.8 | 0.45 |
| Canertinib | 14.1 | 0.67 |
| Ruxolitinib | 12.7 | 0.59 |
| Abrocitinib | 12.6 | 0.58 |
| Bosutinib | 12.3 | 0.55 |
| Abemaciclib | 10.7 | 0.56 |
| Midostaurin | 10.5 | 0.50 |
| Alectinib | 10.4 | 0.65 |
| Fostamatinib | 10.2 | 0.61 |
| Tucatinib | 8.7 | 0.65 |
Known variants
No variants catalogued.