PRKACA
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Capivasertib | 99.7 | 0.64 |
| Netarsudil | 96.6 | 0.68 |
| Baricitinib | 90.9 | 0.62 |
| Midostaurin | 79.8 | 0.50 |
| Ponatinib | 70.9 | 0.53 |
| Ruxolitinib | 45.5 | 0.59 |
| Abrocitinib | 37.8 | 0.58 |
| Darovasertib | 32.9 | 0.72 |
| Pacritinib | 28.8 | 0.45 |
| Defactinib | 23.7 | 0.45 |
| Bosutinib | 22.4 | 0.55 |
| Fostamatinib | 20.9 | 0.61 |
| Brigatinib | 17.2 | 0.51 |
| Gilteritinib | 17.0 | 0.51 |
| Pralsetinib | 15.1 | 0.64 |