Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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PTK2B

RBC: PYK2 · Substrate: pEY + Mn ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Brigatinib99.10.51
Lorlatinib97.60.69
Ponatinib96.40.53
Crizotinib95.10.58
Repotrectinib92.70.61
Ceritinib89.70.62
Defactinib88.00.45
Alectinib85.10.65
Fostamatinib84.90.61
Gilteritinib81.80.51
Sunitinib75.70.52
Bosutinib69.10.55
Entrectinib68.60.67
Pacritinib64.00.45
Midostaurin60.30.50

Known variants

No variants catalogued.
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