SIK2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Bosutinib | 99.6 | 0.55 |
| Nintedanib | 99.4 | 0.61 |
| Midostaurin | 98.8 | 0.50 |
| Brigatinib | 98.4 | 0.51 |
| Dasatinib | 97.5 | 0.70 |
| Fedratinib | 96.8 | 0.58 |
| Pacritinib | 93.0 | 0.45 |
| Vandetanib | 86.8 | 0.72 |
| Dabrafenib | 85.0 | 0.63 |
| Crizotinib | 80.4 | 0.58 |
| Repotrectinib | 76.1 | 0.61 |
| Canertinib | 73.5 | 0.67 |
| Rabusertib | 72.1 | 0.69 |
| Sunitinib | 72.0 | 0.52 |
| Ponatinib | 71.7 | 0.53 |
Known variants
No variants catalogued.