Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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STK11/STRADA/CAB39

RBC: LKB1 · Substrate: LKB1tide ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Pacritinib76.70.45
Repotrectinib68.20.61
Defactinib53.70.45
Pralsetinib35.20.64
Pexidartinib34.40.63
Pazopanib21.20.67
Entrectinib18.30.67
Fostamatinib17.60.61
Netarsudil16.40.68
Quizartinib14.00.74
Canertinib12.80.67
Zanubrutinib11.90.79
Capivasertib11.50.64
Midostaurin10.70.50
Capmatinib10.30.58

Known variants

No variants catalogued.
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