TBK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Midostaurin | 87.1 | 0.50 |
| Pacritinib | 70.8 | 0.45 |
| Nintedanib | 67.1 | 0.61 |
| Fedratinib | 44.1 | 0.58 |
| Bosutinib | 43.8 | 0.55 |
| Sunitinib | 30.3 | 0.52 |
| Axitinib | 30.1 | 0.69 |
| Defactinib | 28.1 | 0.45 |
| Deucravacitinib | 26.0 | 0.72 |
| Abemaciclib | 21.7 | 0.56 |
| Canertinib | 21.6 | 0.67 |
| Entrectinib | 20.5 | 0.67 |
| Fostamatinib | 18.3 | 0.61 |
| Umbralisib | 14.9 | 0.67 |
| Gilteritinib | 14.1 | 0.51 |
Known variants
No variants catalogued.