Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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TESK1

RBC: TESK1 · Substrate: Cofilin 2 + Mn · medium confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Dabrafenib97.00.63
Dasatinib89.80.70
Lorlatinib68.20.69
Repotrectinib66.70.61
Crizotinib50.30.58
Canertinib35.20.67
Ponatinib30.00.53
Erdafitinib26.60.74
Vemurafenib24.10.60
Gilteritinib24.00.51
Everolimus15.80.71
Encorafenib15.50.76
Ruxolitinib15.00.59
Lenvatinib13.40.73
Lapatinib13.10.62

Known variants

No variants catalogued.
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