TYK2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Ruxolitinib | 99.0 | 0.59 |
| Pacritinib | 98.8 | 0.45 |
| Entrectinib | 97.9 | 0.67 |
| Baricitinib | 97.3 | 0.62 |
| Upadacitinib | 97.1 | 0.66 |
| Pralsetinib | 96.8 | 0.64 |
| Repotrectinib | 96.3 | 0.61 |
| Defactinib | 95.0 | 0.45 |
| Fedratinib | 93.6 | 0.58 |
| Midostaurin | 93.4 | 0.50 |
| Abrocitinib | 89.9 | 0.58 |
| Ponatinib | 85.7 | 0.53 |
| Gilteritinib | 85.6 | 0.51 |
| Tofacitinib | 81.0 | 0.68 |
| Nintedanib | 68.7 | 0.61 |
Known variants
No variants catalogued.