VRK2
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Defactinib | 31.4 | 0.45 |
| Bosutinib | 31.3 | 0.55 |
| Lorlatinib | 19.8 | 0.69 |
| Ripretinib | 14.9 | 0.67 |
| Binimetinib | 13.3 | 0.69 |
| Pirtobrutinib | 11.8 | 0.66 |
| Pazopanib | 9.5 | 0.67 |
| Selumetinib | 9.2 | 0.64 |
| Rabusertib | 8.4 | 0.69 |
| Dasatinib | 8.3 | 0.70 |
| Netarsudil | 8.2 | 0.68 |
| Deucravacitinib | 8.0 | 0.72 |
| Mitapivat | 7.6 | 0.63 |
| Zanubrutinib | 7.1 | 0.79 |
| Erdafitinib | 6.8 | 0.74 |
Known variants
No variants catalogued.