Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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ADRBK1

RBC: GRK2 · Substrate: Casein ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Capivasertib19.30.64
Abrocitinib16.10.58
Gilteritinib13.20.51
Quizartinib11.60.74
Canertinib8.60.67
Rabusertib8.50.69
Mitapivat7.60.63
Apatinib6.90.70
Bosutinib6.50.55
Netarsudil5.80.68
Ruxolitinib5.70.59
Axitinib5.70.69
Entrectinib5.20.67
Avapritinib5.20.64
Everolimus5.10.71

Known variants

No variants catalogued.
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