Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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Showing canonical CDK4/CCND1 (URL was CDK4_CYCLIN_D1).
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CDK4/CCND1

RBC: CDK4/cyclin D1 · Substrate: RB Protein ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Abemaciclib99.20.56
Palbociclib99.00.67
Ribociclib94.70.73
Pacritinib86.20.45
Dabrafenib56.70.63
Defactinib37.80.45
Brigatinib34.80.51
Ponatinib28.30.53
Gilteritinib25.10.51
Fedratinib23.80.58
Pirtobrutinib22.20.66
Pemigatinib20.60.72
Avapritinib19.70.64
Crizotinib17.70.58
Infigratinib16.90.71

Known variants

No variants catalogued.
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