CDK8/CCNC
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Midostaurin | 89.0 | 0.50 |
| Brigatinib | 87.0 | 0.51 |
| Sunitinib | 83.1 | 0.52 |
| Abemaciclib | 77.3 | 0.56 |
| Alectinib | 75.3 | 0.65 |
| Bosutinib | 73.3 | 0.55 |
| Baricitinib | 70.0 | 0.62 |
| Ruxolitinib | 69.0 | 0.59 |
| Nintedanib | 68.1 | 0.61 |
| Gilteritinib | 66.2 | 0.51 |
| Ribociclib | 55.6 | 0.73 |
| Palbociclib | 48.8 | 0.67 |
| Lorlatinib | 40.2 | 0.69 |
| Axitinib | 29.1 | 0.69 |
| Capivasertib | 28.7 | 0.64 |
Known variants
No variants catalogued.