DYRK1B
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Abemaciclib | 98.9 | 0.56 |
| Midostaurin | 94.3 | 0.50 |
| Pacritinib | 79.0 | 0.45 |
| Palbociclib | 77.1 | 0.67 |
| Defactinib | 76.1 | 0.45 |
| Alectinib | 68.5 | 0.65 |
| Brigatinib | 65.2 | 0.51 |
| Avapritinib | 47.1 | 0.64 |
| Afatinib | 44.5 | 0.71 |
| Sunitinib | 41.6 | 0.52 |
| Gilteritinib | 41.1 | 0.51 |
| Nintedanib | 35.5 | 0.61 |
| Ruxolitinib | 28.5 | 0.59 |
| Baricitinib | 25.1 | 0.62 |
| Dabrafenib | 24.6 | 0.63 |
Known variants
No variants catalogued.