GRK7
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Repotrectinib | 95.5 | 0.61 |
| Midostaurin | 92.3 | 0.50 |
| Lorlatinib | 92.0 | 0.69 |
| Upadacitinib | 57.2 | 0.66 |
| Capivasertib | 51.8 | 0.64 |
| Darovasertib | 47.1 | 0.72 |
| Defactinib | 25.6 | 0.45 |
| Sunitinib | 25.1 | 0.52 |
| Baricitinib | 20.8 | 0.62 |
| Ceritinib | 13.9 | 0.62 |
| Deucravacitinib | 12.8 | 0.72 |
| Entrectinib | 10.9 | 0.67 |
| Umbralisib | 10.4 | 0.67 |
| Alectinib | 9.8 | 0.65 |
| Pacritinib | 9.8 | 0.45 |
Known variants
No variants catalogued.