IGF1R
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Ceritinib | 98.1 | 0.62 |
| Gilteritinib | 93.4 | 0.51 |
| Brigatinib | 92.0 | 0.51 |
| Entrectinib | 86.5 | 0.67 |
| Fostamatinib | 82.7 | 0.61 |
| Pacritinib | 75.5 | 0.45 |
| Crizotinib | 72.3 | 0.58 |
| Nintedanib | 70.7 | 0.61 |
| Lorlatinib | 67.6 | 0.69 |
| Repotrectinib | 61.6 | 0.61 |
| Osimertinib | 56.9 | 0.73 |
| Defactinib | 50.9 | 0.45 |
| Fedratinib | 49.8 | 0.58 |
| Alectinib | 48.7 | 0.65 |
| Neratinib | 38.6 | 0.60 |
Known variants
No variants catalogued.