Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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MAP2K6

RBC: MKK6 · Substrate: p38a (K53A) ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Encorafenib48.40.76
Pirtobrutinib36.90.66
Lenvatinib36.40.73
Ibrutinib18.70.72
Acalabrutinib17.60.67
Ceritinib16.60.62
Fedratinib16.40.58
Crizotinib15.40.58
Ponatinib15.00.53
Pralsetinib14.50.64
Lapatinib14.20.62
Mobocertinib11.70.76
Remibrutinib10.10.72
Pemigatinib9.90.72
Capmatinib9.40.58

Known variants

No variants catalogued.
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