MARK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Midostaurin | 93.4 | 0.50 |
| Brigatinib | 82.5 | 0.51 |
| Defactinib | 64.2 | 0.45 |
| Axitinib | 58.6 | 0.69 |
| Baricitinib | 54.4 | 0.62 |
| Repotrectinib | 48.8 | 0.61 |
| Sunitinib | 44.6 | 0.52 |
| Pemigatinib | 40.7 | 0.72 |
| Crizotinib | 30.7 | 0.58 |
| Upadacitinib | 29.6 | 0.66 |
| Ruxolitinib | 26.7 | 0.59 |
| Neratinib | 19.9 | 0.60 |
| Pacritinib | 15.9 | 0.45 |
| Bosutinib | 15.5 | 0.55 |
| Canertinib | 13.3 | 0.67 |
Known variants
No variants catalogued.