Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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MAST3

RBC: MAST3 · Substrate: ARPP19 + Mn ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Pacritinib45.50.45
Defactinib35.90.45
Leniolisib18.00.60
Umbralisib16.00.67
Ponatinib14.10.53
Paxalisib12.00.61
Lazertinib11.90.67
Pirtobrutinib11.50.66
Infigratinib11.00.71
Selumetinib10.60.64
Pralsetinib9.90.64
Neratinib8.10.60
Ripretinib7.20.67
Quizartinib6.70.74
Canertinib6.60.67

Known variants

No variants catalogued.
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