Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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NEK1

RBC: NEK1 · Substrate: MBP ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Ponatinib89.90.53
Avapritinib78.70.64
Dabrafenib67.30.63
Erdafitinib65.30.74
Defactinib59.90.45
Pemigatinib59.00.72
Fostamatinib42.60.61
Repotrectinib40.70.61
Neratinib32.70.60
Crizotinib29.60.58
Capivasertib22.90.64
Pacritinib20.30.45
Pazopanib20.00.67
Fedratinib19.90.58
Bosutinib19.80.55

Known variants

No variants catalogued.
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