NEK4
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Ponatinib | 100.0 | 0.53 |
| Defactinib | 81.9 | 0.45 |
| Bosutinib | 76.2 | 0.55 |
| Abemaciclib | 71.4 | 0.56 |
| Gilteritinib | 54.0 | 0.51 |
| Ripretinib | 51.6 | 0.67 |
| Neratinib | 49.9 | 0.60 |
| Brigatinib | 40.0 | 0.51 |
| Crizotinib | 35.5 | 0.58 |
| Repotrectinib | 29.0 | 0.61 |
| Midostaurin | 27.9 | 0.50 |
| Vemurafenib | 22.6 | 0.60 |
| Encorafenib | 21.8 | 0.76 |
| Dabrafenib | 19.9 | 0.63 |
| Pazopanib | 18.9 | 0.67 |
Known variants
No variants catalogued.