NEK5
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Avapritinib | 89.7 | 0.64 |
| Ponatinib | 56.0 | 0.53 |
| Fostamatinib | 52.8 | 0.61 |
| Dabrafenib | 39.8 | 0.63 |
| Pacritinib | 39.0 | 0.45 |
| Pemigatinib | 35.2 | 0.72 |
| Repotrectinib | 34.3 | 0.61 |
| Neratinib | 33.6 | 0.60 |
| Pazopanib | 30.2 | 0.67 |
| Defactinib | 27.0 | 0.45 |
| Pralsetinib | 26.1 | 0.64 |
| Fedratinib | 25.5 | 0.58 |
| Netarsudil | 18.6 | 0.68 |
| Vemurafenib | 17.8 | 0.60 |
| Alpelisib | 16.3 | 0.72 |
Known variants
No variants catalogued.