NEK8
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Lorlatinib | 81.2 | 0.69 |
| Midostaurin | 74.3 | 0.50 |
| Axitinib | 39.9 | 0.69 |
| Ruxolitinib | 30.1 | 0.59 |
| Vemurafenib | 28.1 | 0.60 |
| Baricitinib | 20.0 | 0.62 |
| Lapatinib | 20.0 | 0.62 |
| Bosutinib | 19.8 | 0.55 |
| Dasatinib | 18.9 | 0.70 |
| Fostamatinib | 18.3 | 0.61 |
| Lenvatinib | 17.7 | 0.73 |
| Nilotinib | 17.2 | 0.77 |
| Nintedanib | 16.5 | 0.61 |
| Everolimus | 16.4 | 0.71 |
| Palbociclib | 14.4 | 0.67 |
Known variants
No variants catalogued.