Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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NTRK3

RBC: TRKC · Substrate: pEY ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Pralsetinib99.40.64
Alpelisib99.30.72
Gilteritinib99.00.51
Repotrectinib98.90.61
Entrectinib98.80.67
Larotrectinib98.10.71
Tenalisib98.10.70
Crizotinib97.30.58
Nintedanib96.70.61
Pacritinib96.70.45
Ponatinib96.70.53
Tivozanib96.10.67
Bosutinib95.60.55
Sunitinib95.40.52
Midostaurin95.10.50

Known variants

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