PAK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Neratinib | 82.2 | 0.60 |
| Midostaurin | 43.5 | 0.50 |
| Pralsetinib | 33.1 | 0.64 |
| Fostamatinib | 25.0 | 0.61 |
| Defactinib | 23.9 | 0.45 |
| Pacritinib | 22.1 | 0.45 |
| Bosutinib | 17.6 | 0.55 |
| Ibrutinib | 14.8 | 0.72 |
| Brigatinib | 12.1 | 0.51 |
| Pirtobrutinib | 10.9 | 0.66 |
| Vemurafenib | 10.1 | 0.60 |
| Tenalisib | 10.0 | 0.70 |
| Pazopanib | 9.4 | 0.67 |
| Gedatolisib | 9.2 | 0.61 |
| Osimertinib | 7.4 | 0.73 |
Known variants
No variants catalogued.