Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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SRPK1

RBC: SRPK1 · Substrate: RS peptide · high confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Alectinib99.60.65
Ceritinib50.50.62
Abrocitinib47.90.58
Defactinib35.70.45
Brigatinib24.30.51
Gilteritinib22.90.51
Repotrectinib22.30.61
Midostaurin21.80.50
Lorlatinib19.10.69
Ponatinib14.60.53
Mitapivat14.40.63
Crizotinib14.20.58
Lapatinib13.20.62
Tucatinib11.90.65
Avapritinib11.80.64

Known variants

No variants catalogued.
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