Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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TESK2

RBC: TESK2 · Substrate: Cofilin 2 · medium confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Dasatinib94.40.70
Ponatinib93.60.53
Dabrafenib92.40.63
Encorafenib52.30.76
Regorafenib26.10.72
Pacritinib22.40.45
Sorafenib14.90.78
Ripretinib11.80.67
Imatinib10.80.72
Vemurafenib10.40.60
Dacomitinib9.70.66
Tofacitinib9.30.68
Ceritinib9.00.62
Everolimus8.20.71
Canertinib7.70.67

Known variants

No variants catalogued.
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