VRK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Pacritinib | 53.7 | 0.45 |
| Capivasertib | 25.2 | 0.64 |
| Duvelisib | 24.2 | 0.72 |
| Dabrafenib | 24.0 | 0.63 |
| Encorafenib | 23.5 | 0.76 |
| Abrocitinib | 22.7 | 0.58 |
| Baricitinib | 20.7 | 0.62 |
| Pazopanib | 20.5 | 0.67 |
| Avapritinib | 20.4 | 0.64 |
| Dacomitinib | 20.3 | 0.66 |
| Osimertinib | 20.1 | 0.73 |
| Tofacitinib | 19.7 | 0.68 |
| Fedratinib | 19.5 | 0.58 |
| Tepotinib | 18.6 | 0.73 |
| Mitapivat | 17.5 | 0.63 |
Known variants
No variants catalogued.