Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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WEE1

RBC: WEE1 · Substrate: CDK1 (D146N)/cyclin B1 ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Bosutinib60.00.55
Dasatinib46.10.70
Midostaurin30.30.50
Brigatinib25.80.51
Sunitinib25.70.52
Vemurafenib20.80.60
Gilteritinib19.10.51
Nintedanib18.70.61
Everolimus17.60.71
Netarsudil16.90.68
Acalabrutinib16.50.67
Lapatinib16.20.62
Afatinib16.00.71
Regorafenib15.90.72
Dacomitinib14.40.66

Known variants

No variants catalogued.
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