Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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ARAF

RBC: ARAF · Substrate: MEK1 (K97R) ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Ripretinib100.00.67
Sorafenib100.00.78
Ponatinib99.00.53
Regorafenib98.80.72
Encorafenib97.40.76
Vemurafenib96.90.60
Dabrafenib96.30.63
Apatinib90.70.70
Dasatinib86.20.70
Umbralisib84.90.67
Ibrutinib84.80.72
Nilotinib81.80.77
Upadacitinib64.90.66
Dacomitinib61.50.66
Acalabrutinib58.30.67

Known variants

No variants catalogued.
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