Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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CDK3/CCNE2

RBC: CDK3/cyclin E2 · Substrate: RB Protein ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Defactinib92.00.45
Abemaciclib62.10.56
Pralsetinib58.70.64
Vemurafenib33.00.60
Pacritinib29.00.45
Darovasertib23.20.72
Ponatinib21.00.53
Neratinib19.80.60
Repotrectinib19.70.61
Alectinib17.30.65
Lapatinib16.30.62
Regorafenib16.20.72
Ruxolitinib16.20.59
Midostaurin15.80.50
Pexidartinib14.60.63

Known variants

No variants catalogued.
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