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CDK9/CCNT2

RBC: CDK9/cyclin T2 · Substrate: Pol2-CTD ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Abemaciclib99.00.56
Pacritinib97.90.45
Defactinib91.20.45
Palbociclib84.40.67
Avapritinib54.40.64
Pazopanib49.00.67
Gilteritinib47.70.51
Darovasertib47.40.72
Ribociclib46.50.73
Midostaurin39.10.50
Neratinib31.80.60
Pirtobrutinib31.70.66
Sunitinib30.50.52
Acalabrutinib30.10.67
Abrocitinib29.00.58

Known variants

No variants catalogued.
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