GRK1
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Midostaurin | 86.1 | 0.50 |
| Repotrectinib | 71.1 | 0.61 |
| Lorlatinib | 62.3 | 0.69 |
| Upadacitinib | 38.9 | 0.66 |
| Darovasertib | 37.3 | 0.72 |
| Pirtobrutinib | 23.6 | 0.66 |
| Capivasertib | 21.3 | 0.64 |
| Baricitinib | 18.7 | 0.62 |
| Abemaciclib | 18.6 | 0.56 |
| Pexidartinib | 18.4 | 0.63 |
| Ruxolitinib | 17.3 | 0.59 |
| Quizartinib | 17.2 | 0.74 |
| Neratinib | 15.9 | 0.60 |
| Pralsetinib | 15.5 | 0.64 |
| Sunitinib | 15.1 | 0.52 |
Known variants
No variants catalogued.