PAK3
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Neratinib | 88.3 | 0.60 |
| Midostaurin | 43.0 | 0.50 |
| Defactinib | 40.8 | 0.45 |
| Vemurafenib | 39.9 | 0.60 |
| Pralsetinib | 34.8 | 0.64 |
| Pacritinib | 27.9 | 0.45 |
| Bosutinib | 25.0 | 0.55 |
| Fostamatinib | 20.0 | 0.61 |
| Pirtobrutinib | 19.4 | 0.66 |
| Brigatinib | 13.0 | 0.51 |
| Mobocertinib | 12.8 | 0.76 |
| Fedratinib | 12.7 | 0.58 |
| Gedatolisib | 12.3 | 0.61 |
| Lapatinib | 10.9 | 0.62 |
| Abemaciclib | 10.7 | 0.56 |
Known variants
No variants catalogued.