Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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PAK6

RBC: PAK6 · Substrate: PAKtide ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Pralsetinib41.30.64
Midostaurin38.30.50
Defactinib33.30.45
Axitinib23.80.69
Capivasertib23.50.64
Repotrectinib21.50.61
Avapritinib19.50.64
Brigatinib17.90.51
Darovasertib17.00.72
Neratinib15.50.60
Gilteritinib15.40.51
Baricitinib14.40.62
Canertinib13.00.67
Crizotinib12.60.58
Pacritinib12.50.45

Known variants

No variants catalogued.
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