Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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PKMYT1

RBC: PKMYT1 · Substrate: MBP ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Abemaciclib79.90.56
Alectinib67.20.65
Gilteritinib61.10.51
Palbociclib60.50.67
Midostaurin58.60.50
Sunitinib54.90.52
Vemurafenib49.40.60
Nintedanib47.00.61
Bosutinib44.30.55
Baricitinib40.90.62
Ruxolitinib40.30.59
Regorafenib40.00.72
Netarsudil37.40.68
Afatinib37.00.71
Axitinib36.20.69

Known variants

No variants catalogued.
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