Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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PRKX

RBC: PRKX · Substrate: Kemptide · high confidenceReferenceDerived

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Capivasertib98.30.64
Netarsudil98.30.68
Midostaurin86.10.50
Baricitinib60.20.62
Defactinib53.50.45
Selpercatinib40.60.64
Avapritinib28.50.64
Ponatinib25.70.53
Ruxolitinib23.80.59
Pexidartinib22.80.63
Selumetinib20.00.64
Sunitinib19.80.52
Pacritinib16.10.45
Paxalisib14.20.61
Apatinib13.40.70

Known variants

No variants catalogued.
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