Research Use Only. KIRhub outputs are computational research artifacts. They are not validated for clinical decision-making, diagnosis, or treatment.
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SBK1

RBC: SBK1 · Substrate: PKA sub ·

Top inhibitors

MeasuredDerived
DrugInhibition %Gini
Brigatinib60.40.51
Capivasertib27.10.64
Avapritinib18.00.64
Defactinib16.30.45
Pirtobrutinib13.20.66
Pemigatinib12.50.72
Pacritinib10.70.45
Apatinib9.90.70
Capmatinib9.90.58
Sorafenib9.30.78
Darovasertib9.10.72
Pralsetinib8.80.64
Idelalisib8.40.70
Infigratinib8.30.71
Crizotinib8.10.58

Known variants

No variants catalogued.
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