SIK3
Top inhibitors
| Drug | Inhibition % | Gini |
|---|---|---|
| Dasatinib | 97.8 | 0.70 |
| Midostaurin | 96.4 | 0.50 |
| Bosutinib | 94.9 | 0.55 |
| Pemigatinib | 79.4 | 0.72 |
| Dabrafenib | 72.9 | 0.63 |
| Neratinib | 64.6 | 0.60 |
| Dacomitinib | 55.7 | 0.66 |
| Fedratinib | 49.4 | 0.58 |
| Repotrectinib | 41.9 | 0.61 |
| Brigatinib | 37.8 | 0.51 |
| Erdafitinib | 35.7 | 0.74 |
| Ripretinib | 33.6 | 0.67 |
| Nintedanib | 30.7 | 0.61 |
| Vandetanib | 27.5 | 0.72 |
| Tenalisib | 27.4 | 0.70 |
Known variants
No variants catalogued.